Browsing by Author Reekie, Tristan Andrew

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Showing results 1 to 13 of 13
Issue DateTitleAuthor(s)Citation
2014Body temperature and cardiac changes induced by peripherally administered oxytocin, vaspressin and the non-peptide oxytocin receptor agonist WAY 267, 464: a biotelemetry study in ratsHicks, Callum; Kassiou, Michael; McGregor, Iain; Misagh, G; Narlawar, Rajeshwar; Ramos, Linnet; Reekie, Tristan Andrew; Psychology; Medical Imaging and Radiation Sciences; Psychology; Psychology; Pharmacy; Psychology; Medical Imaging and Radiation SciencesBody temperature and cardiac changes induced by peripherally administered oxytocin, vaspressin and the non-peptide oxytocin receptor agonist WAY 267, 464: a biotelemetry study in rats, British Journal of Pharmacology, vol.171, 11, 2014,pp 2868-2887
2017Comparative evaluation of three TSPO PET radiotracers in a LPS-induced model of mild neuroinflammation in ratsBanister, Samuel; Kassiou, Michael; Reekie, Tristan Andrew; Boutin, Herve; Gerhard, Alexander; Hinz, Rainer; Lepelletier, Francois-Xavier; Sridharan, Sujata; Trigg, William; Medical Radiation Sciences; Chemistry; Medical Imaging and Radiation SciencesComparative evaluation of three TSPO PET radiotracers in a LPS-induced model of mild neuroinflammation in rats, Molecular Imaging and Biology, vol.19, 1, 2017,pp 77-89
2017Discovery and pharmacological evaluation of a novel series of adamantyl cyanoguanidines as P2X7 receptor antagonistsBarron, Melissa; Jackson, Alexander; Kassiou, Michael; McDonnell, Michelle; Munoz, Lenka; O'Brien-Brown, James; Reekie, Tristan Andrew; Schiavini, Paolo; Werry, Eryn; Wilkinson, Shane; Noll, Benjamin D.; Wang, Shudong; School of Medical Sciences: Physiology; Research Grants and Contracts; Chemistry; School of Medical Sciences: Pharmacology; School of Medical Sciences: Pathology; Chemistry; Medical Imaging and Radiation Sciences; Chemistry; Medical Imaging and Radiation Sciences; ChemistryDiscovery and pharmacological evaluation of a novel series of adamantyl cyanoguanidines as P2X7 receptor antagonists, European Journal of Medicinal Chemistry, vol.130, N/A, 2017,pp 433-439
2016Flexible analogues of WAY-267,464: Synthesis and pharmacology at the human oxytocin and vasopressin 1a receptorsGulliver, Damien; Jorgensen, William Thomas; Kassiou, Michael; Reekie, Tristan Andrew; Werry, Eryn; Connor, Mark; School of Medical Sciences: Pharmacology; Chemistry; Medical Imaging and Radiation Sciences; Medical Imaging and Radiation Sciences; Medical Imaging and Radiation SciencesFlexible analogues of WAY-267,464: Synthesis and pharmacology at the human oxytocin and vasopressin 1a receptors, European Journal of Medicinal Chemistry, vol.108, N/A, 2016,pp 730-740
2016The Formation of Seven-Membered Heterocycles under Mild Pictet-Spengler Conditions: A Route to Pyrazolo[3,4]benzodiazepinesJorgensen, William Thomas; Kassiou, Michael; Katte, Timothy; Reekie, Tristan Andrew; Chemistry; Chemistry; Chemistry; Medical Imaging and Radiation SciencesThe Formation of Seven-Membered Heterocycles under Mild Pictet-Spengler Conditions: A Route to Pyrazolo[3,4]benzodiazepines, The Journal of Organic Chemistry, vol.81, 11, 2016,pp 4883-4889
2017Investigation of pyrazolo-sulfonamides as putative small molecule oxytocin receptor agonistsGulliver, Damien; Jorgensen, William Thomas; Kassiou, Michael; Katte, Timothy; Reekie, Tristan Andrew; Werry, Eryn; Wong, Erick; Boyd, Rochelle; Connor, Mark; School of Medical Sciences: Pharmacology; Chemistry; Chemistry; Chemistry; Medical Imaging and Radiation Sciences; Medical Imaging and Radiation Sciences; School of Medical Sciences: PharmacologyInvestigation of pyrazolo-sulfonamides as putative small molecule oxytocin receptor agonists, European Journal of Medicinal Chemistry, vol.136, N/A, 2017,pp 330-333
2014Investigations of amide bond variation and biaryl modification in analogues of alpha7 nAChR agonist SEN12333Beinat, Corinne; Hibbs, David; Kassiou, Michael; Reekie, Tristan Andrew; Coles, Carolyn; Harvey, Andrew; O'Connor, Susan; Olson, Thao T.; Tsanaktsidis, John; Xiao, Yingxian; Xie, Teresa; Chemistry; Pharmacy; Medical Imaging and Radiation Sciences; Medical Imaging and Radiation SciencesInvestigations of amide bond variation and biaryl modification in analogues of alpha7 nAChR agonist SEN12333, European Journal of Medicinal Chemistry, vol.84, N/A, 2014,pp 200-205
2014Pyrazolo 1,4 diazepines as non-peptidic probes of the oxytocin and vasopressin receptorsKassiou, Michael; McGregor, Iain; Reekie, Tristan Andrew; Medical Imaging and Radiation Sciences; Psychology; Medical Imaging and Radiation SciencesPyrazolo 1,4 diazepines as non-peptidic probes of the oxytocin and vasopressin receptors, Tetrahedron Letters, vol.55, 33, 2014,pp 4568-4571
2017Rapid access to N-(indol-2-yl)amides and N-(indol-3-yl)amides as unexplored pharmacophoresHibbs, David; Kassiou, Michael; Law, Vivian; Ong, Jennifer; Reekie, Tristan Andrew; Wilkinson, Shane; Pharmacy; Chemistry; Chemistry; Pharmacy; Medical Imaging and Radiation Sciences; ChemistryRapid access to N-(indol-2-yl)amides and N-(indol-3-yl)amides as unexplored pharmacophores, Organic and Biomolecular Chemistry, vol.15, 3, 2017,pp 576-580
2017Ring-opened aminothienopyridazines as novel tau aggregation inhibitorsKassiou, Michael; Moir, Michael; Reekie, Tristan Andrew; Chua, Sook Wern; Ittner, Arne; Ittner, Lars; Martin, Andrew; Chemistry; Chemistry; Medical Imaging and Radiation SciencesRing-opened aminothienopyridazines as novel tau aggregation inhibitors, MedChemComm (Medicinal Chemistry Communications), vol.8, 6, 2017,pp 1275-1282
2017Structural optimization and pharmacological evaluation of inhibitors targeting dual-specificity tyrosine phosphorylation-regulated kinases (DYRK) and CDC-like kinases (CLK) inglioblastomaAbbassi, Ramzi; Font Sadurni, Josep; Hoque, Monira; Kassiou, Michael; Munoz, Lenka; Phoa, Athena; Reekie, Tristan Andrew; Ryan, Renae; Zhou, Qingdi; Day, Bryan W.; Johns, Terrance G; Stringer, Brett W.; School of Medical Sciences: Pharmacology; School of Molecular Bioscience (SMB); Pharmacy; Chemistry; School of Medical Sciences: Pathology; School of Medical Sciences: Pharmacology; Medical Imaging and Radiation Sciences; School of Medical Sciences: Pharmacology; ChemistryStructural optimization and pharmacological evaluation of inhibitors targeting dual-specificity tyrosine phosphorylation-regulated kinases (DYRK) and CDC-like kinases (CLK) inglioblastoma, Journal of Medicinal Chemistry, vol.60, 5, 2017,pp 2052-2070
2015Structure-activity relationship studies of SEN12333 analogues: Determination of the optimal requirements for binding affinities at alpha7 nAChRs through incorporation of known structural motifsBeinat, Corinne; Kassiou, Michael; O'Brien-Brown, James; Reekie, Tristan Andrew; Banister, Samuel D.; Coles, Carolyn; Grishin, Anton; Harvey, Andrew; Kolesik, Peter; OConnor, Susan; Olson, Thao T.; Tsanaktsidis, John; Xiao, Yingxian; Xie, Teresa; Chemistry; Medical Imaging and Radiation Sciences; Chemistry; Medical Imaging and Radiation SciencesStructure-activity relationship studies of SEN12333 analogues: Determination of the optimal requirements for binding affinities at alpha7 nAChRs through incorporation of known structural motifs, European Journal of Medicinal Chemistry, vol.95, N/A, 2015,pp 277-301
2016A systematic exploration of the effects of flexibility and basicity on sigma (sigma) receptor binding in a series of substituted diaminesConroy, Trent; Gong, Yu; Kassiou, Michael; Manohar, Madhura; Reekie, Tristan Andrew; Rendina, Louis; Webster, Michael William; Wilkinson, Shane; Banister, Samuel D.; Lieberman, Brian P.; Mach, Robert H.; Chemistry; Chemistry; Chemistry; Chemistry; Medical Imaging and Radiation Sciences; Chemistry; Molecular Bioscience; ChemistryA systematic exploration of the effects of flexibility and basicity on sigma (sigma) receptor binding in a series of substituted diamines, Organic and Biomolecular Chemistry, vol.14, 39, 2016,pp 9388-9405