Browsing by Author Jensen, Anders

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Showing results 1 to 11 of 11
Issue DateTitleAuthor(s)Citation
20145-(Piperidin-4-yl)-3-Hydroxypyrazole: A Novel Scaffold for Probing the Orthosteric gamma-Aminobutyric Acid Type A Receptor Binding SiteBalle, Thomas; Sorensen, Troels; Frolund, Bente; Jensen, Anders; Kongstad, Kenneth T; Krall, Jacob; Nielsen, Birgitte; Pharmacy; Pharmacy5-(Piperidin-4-yl)-3-Hydroxypyrazole: A Novel Scaffold for Probing the Orthosteric gamma-Aminobutyric Acid Type A Receptor Binding Site, ChemMedChem: chemistry enabling drug discovery, vol.9, 11, 2014,pp 2475-2485
2015Conformationally restrained carbamoylcholine homologues. Synthesis, pharmacology at neuronal nicotinic acetylcholine receptors and biostructural considerationsBalle, Thomas; De La Fuente Revenga, Mario; Frølund, Bente; Jensen, Anders; PharmacyConformationally restrained carbamoylcholine homologues. Synthesis, pharmacology at neuronal nicotinic acetylcholine receptors and biostructural considerations, European Journal of Medicinal Chemistry, vol.102, N/A, 2015,pp 352-362
2013Design, Synthesis, and Biological Evaluation of Erythrina Alkaloid Analogues as Neuronal Nicotinic Acetylcholine Receptor AntagonistsBalle, Thomas; Andersen, Jacob; Andreasen, Jesper; Borch, Morten; Crestey, Francois; Jensen, Anders; Kristensen, Jesper; PharmacyDesign, Synthesis, and Biological Evaluation of Erythrina Alkaloid Analogues as Neuronal Nicotinic Acetylcholine Receptor Antagonists, Journal of Medicinal Chemistry, vol.56, 23, 2013,pp 9673-9682
2015Exploration of the molecular architecture of the orthosteric binding site in the alpha4beta2 nicotinic acetylcholine receptor with analogs of 3-(dimethylamino)butyl dimethylcarbamate (DMABC) and 1-(pyridin-3-yl)-1,4-diazepaneBalle, Thomas; Liu, Jun; Sorensen, Troels; Bach, Tinna; Blaazer, Antoni; Della Volpe, Serena; Frolund, Bente; Jensen, Anders; Petersen, Jette; Van Muijlwijk-Koezen, Jacqueline; Pharmacy; Pharmacy; PharmacyExploration of the molecular architecture of the orthosteric binding site in the alpha4beta2 nicotinic acetylcholine receptor with analogs of 3-(dimethylamino)butyl dimethylcarbamate (DMABC) and 1-(pyridin-3-yl)-1,4-diazepane, European Journal of Medicinal Chemistry, vol.102, N/A, 2015,pp 425-444
2013Exploring the Orthosteric Binding Site of the y-Aminobutyric Acid Type A Receptor Using 4-(Piperidin-4-yl)-1-hydroxypyrazoles 3- or 5-Imidazolyl Substituted: Design, Synthesis, and Pharmacological EvaluationBalle, Thomas; Sorensen, Troels; Frolund, Bente; Jensen, Anders; Jensen, Claus H; Krall, Jacob; Nielsen, Birgitte; Sander, Tommy; Pharmacy; PharmacyExploring the Orthosteric Binding Site of the y-Aminobutyric Acid Type A Receptor Using 4-(Piperidin-4-yl)-1-hydroxypyrazoles 3- or 5-Imidazolyl Substituted: Design, Synthesis, and Pharmacological Evaluation, Journal of Medicinal Chemistry, vol.56, 16, 2013,pp 6536-6540
2016Kavain, the Major Constituent of the Anxiolytic Kava Extract, Potentiates GABAA Receptors: Functional Characteristics and Molecular MechanismAbsalom, Nathan Luke; Christensen, Emilie; Chua, Han Chow; Collins, Mary; Hartiadi, Leonny Yulita; Ramzan, Iqbal; Hoestgaard-Jensen, Kirsten; Jensen, Anders; Pharmacy; Pharmacy; Pharmacy; Pharmacy; Pharmacy; PharmacyKavain, the Major Constituent of the Anxiolytic Kava Extract, Potentiates GABAA Receptors: Functional Characteristics and Molecular Mechanism, PloS One, vol.11, 6, 2016,pp 1-17
2016Kavain, the Major Constituent of the Anxiolytic Kava Extract, Potentiates GABAA Receptors: Functional Characteristics and Molecular MechanismAbsalom, Nathan Luke; Christensen, Emilie; Chua, Han Chow; Collins, Mary; Hartiadi, Leonny Yulita; Ramzan, Iqbal; Hoestgaard-Jensen, Kirsten; Jensen, Anders; Pharmacy; Pharmacy; Pharmacy; Pharmacy; Pharmacy; PharmacyKavain, the Major Constituent of the Anxiolytic Kava Extract, Potentiates GABAA Receptors: Functional Characteristics and Molecular Mechanism, PloS One, vol.11, 6, 2016,pp 1-17
2013Synthesis and biological evaluation of 4-(aminomethyl)-1-hydroxypyrazole analogues of muscimol as I?-aminobutyric acid(a) receptor agonistsBalle, Thomas; Bergmann, Rikke; Frølund, Bente; Frydenvang, Karla; Jensen, Anders; Jogensen, Charlotte; Kehler, Jan; Kristensen, Jesper; Kristiansen, Uffe; Moller, Henriette A; Nielsen, Birgitte; Petersen, Jette; PharmacySynthesis and biological evaluation of 4-(aminomethyl)-1-hydroxypyrazole analogues of muscimol as I?-aminobutyric acid(a) receptor agonists, Journal of Medicinal Chemistry, vol.56, 3, 2013,pp 993-1006
2014Synthesis and pharmacological evaluation of 6-aminonicotinic acid analogues as novel GABAA receptor agonistsBalle, Thomas; Soerensen, Troels; Bergmann, Rikke; Damgaard, Maria; Frølund, Bente; Jensen, Anders; Nielsen, Birgitte; Petersen, Jette; Pharmacy; PharmacySynthesis and pharmacological evaluation of 6-aminonicotinic acid analogues as novel GABAA receptor agonists, European Journal of Medicinal Chemistry, vol.84, N/A, 2014,pp 404-416
2013Synthesis, pharmacology, and biostructural characterization of novel alpha4beta2 nicotinic acetylcholine receptor agonistsBalle, Thomas; Ahring, Philip; Frølund, Bente; Gajhede, Michael; Hansen, Camilla P; Jensen, Anders; Kastrup, Jette Sandholm; Nielsen, Elsebet; Petersen, Jette; Rohde, Line Aagot Hede; Ussing, Christine; PharmacySynthesis, pharmacology, and biostructural characterization of novel alpha4beta2 nicotinic acetylcholine receptor agonists, Journal of Medicinal Chemistry, vol.56, 3, 2013,pp 940-951
2015Tying up Nicotine: New Selective Competitive Antagonist of the Neuronal Nicotinic Acetylcholine ReceptorsBalle, Thomas; Indurthi Venkata, Dinesh; Andreasen, Jesper; Crestey, Francois; Jensen, Anders; Kristensen, Jesper; Pedersen, Henrik; Petersen, Ida; Pharmacy; PharmacyTying up Nicotine: New Selective Competitive Antagonist of the Neuronal Nicotinic Acetylcholine Receptors, ACS Medicinal Chemistry Letters, vol.6, 4, 2015,pp 472-475