Browsing by Author Dolle, Frederic

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Issue DateTitleAuthor(s)Citation
200711C-DPA-713: A novel peripheral benzodiazepine receptor PET ligand for in vivo imaging of neuroinflammationKassiou, Michael; Boutin, Herve; Chauveau, Fabien; Dolle, Frederic; Gregoire, Marie-Claude; Hantraye, Philippe; James, Michelle L; Tavitian, Bertrand; Thominiaux, Cyrille; Trebossen, Regine; Medical Radiation Sciences11C-DPA-713: A novel peripheral benzodiazepine receptor PET ligand for in vivo imaging of neuroinflammation, The Journal of Nuclear Medicine, vol.48,(4),2007,pp 573-581
200918F-ZW-104: A new radioligand for imaging neuronal nicotinic acetylcholine receptors - In vitro binding properties and PET studies in baboonsKassiou, Michael; Bottlaender, Michael; Damont, Annelaure; Dolle, Frederic; Kellar, Kenneth J; Kosikowski, Alan; Schollhorn-Peyronneau, Marie-Anne; Valette, Heric; Wei, Zhi-Liang; Xiao, Yingxian; Medical Imaging and Radiation Sciences18F-ZW-104: A new radioligand for imaging neuronal nicotinic acetylcholine receptors - In vitro binding properties and PET studies in baboons, The Journal of Nuclear Medicine, vol.50, 8,pp 1349-1355
2014[18F]DPA-C5yne, a novel fluorine-18-labelled analogue of DPA-714: radiosynthesis and preliminary evaluation as a radiotracer for imaging neuroinflammation with PETKassiou, Michael; Bernards, Nicholas; Boisgard, Raphael; Damont, Annelaure; Dolle, Frederic; Kuhnast, Bertrand; Marguet, Frank; Medran-Navarrete, Vincent; Peyronneau, Marie-Anne; Pottier, Geraldine; Puech, Frederic; Medical Imaging and Radiation Sciences[18F]DPA-C5yne, a novel fluorine-18-labelled analogue of DPA-714: radiosynthesis and preliminary evaluation as a radiotracer for imaging neuroinflammation with PET, Journal of Labelled Compounds and Radiopharmaceuticals, vol.57, 6, 2014,pp 410-418
2007Acetylenic pyridines for use in PET imaging of nicotinic receptorsFulton, Roger; Henderson, David; Kassiou, Michael; Chellappan, Sheela K; Dolle, Frederic; Emond, Patrick; Giboureau, Nicolas; Guilloteau, Denis; Kellar, Kenneth J; Kozikowski, Alan P; Wei, Zhi-Liang; Xiao, Yingxian; Physics; Medicine; Medical Radiation SciencesAcetylenic pyridines for use in PET imaging of nicotinic receptors, ChemMedChem: chemistry enabling drug discovery, vol.2,(0),2007,pp 54-57
2009Comparative evaluation of the translocator protein radioligands (11)C-DPA-713, (18)F-DPA-714, and (11)C-PK11195 in a rat model of acute neuroinflammationJames, Michelle; Kassiou, Michael; Boutin, Herve; Chauveau, Fabien; Damont, Annelaure; Dolle, Frederic; Hinnen, Francoise; Kuhnast, B; Tavitian, Bertrand; Van Camp, Nadja; School of Medical Sciences: Pharmacology; Medical Radiation SciencesComparative evaluation of the translocator protein radioligands (11)C-DPA-713, (18)F-DPA-714, and (11)C-PK11195 in a rat model of acute neuroinflammation, The Journal of Nuclear Medicine, vol.50,(3),2009,pp 468-476
2008Dopamine D1 Receptor Imaging in the Rodent and Primate Brain Using the Isoquinoline (+)-[(11)C]A-69024 and Positron Emission TomographyKassiou, Michael; Besret, Laurent; Bottlaender, Michel; Coulon, Christine; Demphel, Stephane; Dolle, Frederic; Guillermier, Martine; Hantraye, Philippe; Herard, Anne-Sophie; Hinnen, Francoise; Ottaviani, Michelle; Medical Imaging and Radiation SciencesDopamine D1 Receptor Imaging in the Rodent and Primate Brain Using the Isoquinoline (+)-[(11)C]A-69024 and Positron Emission Tomography, Journal of Pharmaceutical Sciences, vol.97, 7, 2008,pp 2811-2819
2007DPA-714 A new translocator protein (18kDa) ligand: Synthesis, radiofluorination and pharmacological characterisationJames, Michelle; Kassiou, Michael; Chalon, Sylvie; Dolle, Frederic; Eberl, Stefan; Fulton, Roger R.; Garreau, Lucette; Guilloteau, Denis; Henderson, David J.; Selleri, Silvia; Vercouille, J; School of Medical Sciences: Pharmacology; Medical Radiation SciencesDPA-714 A new translocator protein (18kDa) ligand: Synthesis, radiofluorination and pharmacological characterisation, N/A, vol.50,(),2007,pp N/A-N/A
2008DPA-714, a New Translocator Protein-Specific Ligand: Synthesis, Radiofluorination, and Pharmacologic CharacterizationJames, Michelle; Kassiou, Michael; Chalon, Sylvie; Dolle, Frederic; Fulton, Roger R.; Garreau, Lucette; Guilloteau, Denis; Henderson, David J.; Selleri, Silvia; Vercoullie, Johnny; School of Medical Sciences: Pharmacology; Medical Imaging and Radiation SciencesDPA-714, a New Translocator Protein-Specific Ligand: Synthesis, Radiofluorination, and Pharmacologic Characterization, The Journal of Nuclear Medicine, vol.49, 5, 2008,pp 814-822
2010Evaluation of the PBR/TSPO radioloigand [18F]DPA-714 in a rat model of focal cerebral ischemiaKassiou, Michael; Abraham, Martin; Boisgard, R; Damont, Annelaure; Dolle, Frederic; Kuhnast, Bertrand; Tavitian, Bertrand; Theze, Benoit; Van Camp, Nadja; Medical Imaging and Radiation SciencesEvaluation of the PBR/TSPO radioloigand [18F]DPA-714 in a rat model of focal cerebral ischemia, Journal of Cerebral Blood Flow and Metabolism, vol.30, 1, 2010,pp 230-241
2010Fluorine-18 chemistry for PET: A concise introductionBanister, Samuel; Kassiou, Michael; Dolle, Frederic; Roeda, Dirk; Chemistry; Medical Imaging and Radiation SciencesFluorine-18 chemistry for PET: A concise introduction, Current Radiopharmaceuticals, vol.3, 2,pp 68-80
2006Improved synthesis of the peripheral benzodiazepine receptor ligand C-11 DPA-713 using C-11 methyl triflate.James, Michelle; Kassiou, Michael; Besret, Laurent; Bottlaender, Michel; Boutin, Herve; Bramoulle, Yann; Dolle, Frederic; Gregoire, M. C.; Hantraye, Ph; Selleri, Silvia; Tavitian, Bertrand; Thominiaux, Cyrille; Valette, Heric; School of Medical Sciences: Pharmacology; Medical Radiation SciencesImproved synthesis of the peripheral benzodiazepine receptor ligand C-11 DPA-713 using C-11 methyl triflate., Applied Radiation and Isotopes, vol.64,(5),2006,pp 570-573
2013Metabolism and quantification of [(18)F]DPA-714, a new TSPO positron emission tomography radioligandKassiou, Michael; Bottlaender, Michael; Damont, Annelaure; Dolle, Frederic; Goutal, Sebastien; Saba, W; Schollhorn-Peyronneau, Marie-Anne; Valette, Heric; Medical Imaging and Radiation SciencesMetabolism and quantification of [(18)F]DPA-714, a new TSPO positron emission tomography radioligand, Drug Metabolism and Disposition, vol.41, 1, 2013,pp 122-131
2002Preparation of a bromine-76 labelled analogue of epibatidine: a potent ligand for nicotinic acetylcholine receptor studiesKassiou, Michael; Crouzel, C.; Dannals, Robert F.; Dolci, L.; Dolle, Frederic; Loc'h, Christian; Maziere, Bernard; Musachio, John L.; Medical Radiation SciencesPreparation of a bromine-76 labelled analogue of epibatidine: a potent ligand for nicotinic acetylcholine receptor studies, Applied Radiation and Isotopes, vol.57,(5),2002,pp 713-717
2010Pyrazolo[1,5-a]pyrimidine acetamides: 4-Phenyl alkyl ether derivatives as potent ligands for the 18 kDa translocator protein (TSPO)Hanani, Raphy; Hibbs, David; Kassiou, Michael; Reynolds, Aaron; Da Pozzo, Eleonora; Damont, Annelaure; Dolle, Frederic; Martini, Claudia; Selleri, Silvia; Chemistry; Pharmacy; Medical Radiation Sciences; ChemistryPyrazolo[1,5-a]pyrimidine acetamides: 4-Phenyl alkyl ether derivatives as potent ligands for the 18 kDa translocator protein (TSPO), Bioorganic & Medicinal Chemistry Letters: the tetrahedron journal for research at the interface of chemistry and biology, vol.20, 19,pp 5799-5802
2009Radiolabelled molecules for imaging the translocator protein (18 kDa) using positron emission tomographyKassiou, Michael; Luus, Christopher; Reynolds, Aaron; Dolle, Frederic; Medical Radiation Sciences; School of Medical Sciences: Pharmacology; ChemistryRadiolabelled molecules for imaging the translocator protein (18 kDa) using positron emission tomography, Current Medicinal Chemistry, vol.16,(22),2009,pp 2899-2923
2004Radiosynthesis And In Vivo Evaluation Of [11C]Ro-547312: A Novel Nr1/2B Subtype Selective Nmda Receptor RadioligandKassiou, Michael; Bottlaender, Michel; Coulon, Christine; Demphel, Stephane; Dolle, Frederic; Ottaviani, Michelle; Valette, Heric; Medical Radiation SciencesRadiosynthesis And In Vivo Evaluation Of [11C]Ro-547312: A Novel Nr1/2B Subtype Selective Nmda Receptor Radioligand, Journal of Labelled Compounds and Radiopharmaceuticals, vol.47,(13),2004,pp 911-920
2004Radiosynthesis And Pharmacological Evaluation Of [11C]Emd-95885: A High Affinity Ligand For Nr2B-Containing Nmda Receptors.Kassiou, Michael; Liu, Xiang; Besret, Laurent; Bottlaender, Michel; Bramoulle, Yann; Coulon, Christine; de Bruin, Beatrice; Dolle, Frederic; Ottaviani, Michelle; Roger, Gaelle; Valette, Heric; Medical Radiation Sciences; School of Medical Sciences: PharmacologyRadiosynthesis And Pharmacological Evaluation Of [11C]Emd-95885: A High Affinity Ligand For Nr2B-Containing Nmda Receptors., Bioorganic & Medicinal Chemistry, vol.12,(12),2004,pp 3229-3237
2007Radiosynthesis and preliminary evaluation of ZW-90 and ZW-110, two novel acetylenic pyridines for imaging nicotonic receptorsFulton, Roger; Henderson, David; Kassiou, Michael; Chellappan, Sheela K; Dolle, Frederic; Emond, Patrick; Giboureau, Nicolas; Guilloteau, Denis; Kellar, Kenneth J; Kozikowski, Alan P; Wei, Zhi-Liang; Xiao, Yingxian; Physics; Medicine; Medical Radiation SciencesRadiosynthesis and preliminary evaluation of ZW-90 and ZW-110, two novel acetylenic pyridines for imaging nicotonic receptors, N/A, vol.N/A,(),2007,pp N/A-N/A
2006Radiosynthesis of (E)-N-(2- C-11 methoxybenzyl)-3-phenyl-acrylamidine, a novel subnanomolar NR2B subtype-selective NMDA receptor antagonist.Kassiou, Michael; Besret, Laurent; Bottlaender, Michel; Bramoulle, Yann; de Bruin, Beatrice; Demphel, Stephane; Dolle, Frederic; Hinnen, Francoise; Thominiaux, Cyrille; Valette, Heric; Medical Radiation SciencesRadiosynthesis of (E)-N-(2- C-11 methoxybenzyl)-3-phenyl-acrylamidine, a novel subnanomolar NR2B subtype-selective NMDA receptor antagonist., Applied Radiation and Isotopes, vol.64,(3),2006,pp 348-354
2008Radiosynthesis of [(18)F]DPA-714, a selective radioligand for imaging the translocator protein (18 kDa) PETJames, Michelle; Kassiou, Michael; Luus, Christopher; Damont, Annelaure; Dolle, Frederic; Hinnen, Francoise; Kuhnast, B; Schollhorn-Peyronneau, Marie-Anne; Tavitian, Bertrand; School of Medical Sciences: Pharmacology; Medical Imaging and Radiation Sciences; School of Medical Sciences: PharmacologyRadiosynthesis of [(18)F]DPA-714, a selective radioligand for imaging the translocator protein (18 kDa) PET, Journal of Labelled Compounds and Radiopharmaceuticals, vol.51, 7-8, 2008,pp 286-292